imveliso

Ixabiso elihle I-Pharmaceutical intermediates 99% Nicergoline CAS 27848-84-6

Inkcazelo emfutshane:


Iinkcukacha zeMveliso

Iithegi zeMveliso

Ingcaciso yeMveliso

Ixabiso elihle I-Pharmaceutical intermediates 99% Nicergoline CAS 27848-84-6

Iinkcukacha zeMveliso:
Igama leKhemikhali: Nicergoline

Ifomula yemolekyuli:C24H26BrN3O3

Inombolo yeCAS: 27848-84-6

IBakala: CP/EP/USP

Ezinye iiNkcazelo eziNxulumeneyo

Intshayelelo:
Nicergoline, njengoko Sermion, Joseph Hermione, nicergoline, Kell; uphumelele i-ninni cabergoline chemical yokuqala ebizwa ngokuba yi-alpha 10 methoxy two methyl -1,6- cabergoline -8 beta 5''- nicotinate. I-Bromine methanol esekelwe kwifomula yemolekyuli: c24h26brn3o3 ubunzima bemolekyuli yi-484.39. okanye izibonakaliso ezibukhali zokuphazamiseka kwengqondo okungapheliyo okanye ukungasebenzi kakuhle kwe-cerebral metabolic. Ukushukuma, ukungasebenzi kakuhle kwengqondo okubangelwa yimiqobo yolwimi, isiyezi, i-tinnitus, ukubona luzizi, ukuziva, intloko ebuhlungu, ukuphuthelwa, ukulahleka kwenkumbulo, ukungakhathali, ukudakumba, ukuxhalaba, imincili kunye nokuphazamiseka kwengqondo. I-Nicergoline Tablets inokonyusa uxinzelelo lwegazi ukusebenza kweziyobisi. Ngenxa ye-nicergoline i-metabolized yi-CytochromeP4502D6, ayibandakanyi ukusebenzisana neziyobisi ngendlela efanayo.

Imisebenzi:
1. I-Nicergoline yi-ergot derivative esetyenziselwa ukunyanga i-senile dementia kunye nezinye iziphazamiso ezinemvelaphi ye-vascular.

2. Kufunyaniswe ukuba yonyusa amandla engqondo kunye nokwandisa ukucaca kunye nokuqonda.

3. Yehlisa ukuxhathisa kwemithambo kwaye yonyusa ukuhamba kwegazi kwi-arterial ebuchosheni, iphucula ukusetyenziswa kweoksijini kunye neglucose ziiseli zengqondo.

4. Ineempawu ezifanayo ze-vasoactive kwezinye iindawo zomzimba, ngakumbi imiphunga.

5. Isetyenziselwa ukuphazamiseka kwemithambo yegazi efana ne-cerebral thrombosis kunye ne-atherosclerosis, i-arterial blockages kwimilenze, isifo sikaRaynaud, i-vascular migraines, kunye ne-retinopathy.

6. I-Nicergoline ibhaliswe kumazwe angaphezu kwamashumi amahlanu kwaye isetyenziswe iminyaka engaphezu kwamashumi amathathu kunyango lwengqondo, i-affective, kunye nokuziphatha kwabantu abadala.

Ukupakisha:
ingxowa yeplastiki ngaphakathi kunye nebhegi ye-aluminiyam ngaphandle
Ugcino :Emthunzini wobumnyama kunye nemeko. Kwaye ubushushu obuphantsi (+2-+8ºC)

Inkcazo

INTO
INDEX
Iimpawu
Ikristale emhlophe okanye umgubo
Indawo yokunyibilika
133ºC ~ 136ºC
Ukujikeleza okuthe ngqo
Iyahambelana
Ukucaca kunye nombala wesisombululo
Cacileyo
Izinto ezinxulumeneyo
Ukungcola ngokupheleleyo ≤1.5%
Nor-nocergoline (B) ≤0.50%
I-Chioronicergoline (A) ≤0.5%
I-MeLUOL (C) ≤0.30%
Ukungcola okungachazwanga: ≤0.30%
Amanzi
≤0.5%
Intsimbi enzima
≤20ppm
Intsalela ekutshisweni
≤0.05%
Isivavanyi
98.5%~102%
Izinyibilikisi ezishiyekileyo
I-acetone
≤1000ppm
Diethyl ether
≤2000ppm
I-Ethanol
≤1000ppm
IMethanol
≤1000ppm
Toluene
≤500ppm
IDichloromethan
≤100ppm
I-Triethylamine
≤500ppm
Ukuqukumbela
Ukuhambelana ne-EP 5.0
* Ukongeza: Inkampani inokuphanda kwaye iphuhlise iimveliso ezintsha ngokwemfuno ekhethekileyo yabathengi bethu.

 


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