Ixabiso elihle I-Pharmaceutical intermediates 99% Nicergoline CAS 27848-84-6
Ixabiso elihle I-Pharmaceutical intermediates 99% Nicergoline CAS 27848-84-6
Iinkcukacha zeMveliso:
Igama leKhemikhali: Nicergoline
Ifomula yemolekyuli:C24H26BrN3O3
Inombolo yeCAS: 27848-84-6
IBakala: CP/EP/USP
Intshayelelo:
Nicergoline, njengoko Sermion, Joseph Hermione, nicergoline, Kell; uphumelele i-ninni cabergoline chemical yokuqala ebizwa ngokuba yi-alpha 10 methoxy two methyl -1,6- cabergoline -8 beta 5''- nicotinate. I-Bromine methanol esekelwe kwifomula yemolekyuli: c24h26brn3o3 ubunzima bemolekyuli yi-484.39. okanye izibonakaliso ezibukhali zokuphazamiseka kwengqondo okungapheliyo okanye ukungasebenzi kakuhle kwe-cerebral metabolic. Ukushukuma, ukungasebenzi kakuhle kwengqondo okubangelwa yimiqobo yolwimi, isiyezi, i-tinnitus, ukubona luzizi, ukuziva, intloko ebuhlungu, ukuphuthelwa, ukulahleka kwenkumbulo, ukungakhathali, ukudakumba, ukuxhalaba, imincili kunye nokuphazamiseka kwengqondo. I-Nicergoline Tablets inokonyusa uxinzelelo lwegazi ukusebenza kweziyobisi. Ngenxa ye-nicergoline i-metabolized yi-CytochromeP4502D6, ayibandakanyi ukusebenzisana neziyobisi ngendlela efanayo.
Imisebenzi:
1. I-Nicergoline yi-ergot derivative esetyenziselwa ukunyanga i-senile dementia kunye nezinye iziphazamiso ezinemvelaphi ye-vascular.
2. Kufunyaniswe ukuba yonyusa amandla engqondo kunye nokwandisa ukucaca kunye nokuqonda.
3. Yehlisa ukuxhathisa kwemithambo kwaye yonyusa ukuhamba kwegazi kwi-arterial ebuchosheni, iphucula ukusetyenziswa kweoksijini kunye neglucose ziiseli zengqondo.
4. Ineempawu ezifanayo ze-vasoactive kwezinye iindawo zomzimba, ngakumbi imiphunga.
5. Isetyenziselwa ukuphazamiseka kwemithambo yegazi efana ne-cerebral thrombosis kunye ne-atherosclerosis, i-arterial blockages kwimilenze, isifo sikaRaynaud, i-vascular migraines, kunye ne-retinopathy.
6. I-Nicergoline ibhaliswe kumazwe angaphezu kwamashumi amahlanu kwaye isetyenziswe iminyaka engaphezu kwamashumi amathathu kunyango lwengqondo, i-affective, kunye nokuziphatha kwabantu abadala.
Ukupakisha:
ingxowa yeplastiki ngaphakathi kunye nebhegi ye-aluminiyam ngaphandle
Ugcino :Emthunzini wobumnyama kunye nemeko. Kwaye ubushushu obuphantsi (+2-+8ºC)
INTO | INDEX |
Iimpawu | Ikristale emhlophe okanye umgubo |
Indawo yokunyibilika | 133ºC ~ 136ºC |
Ukujikeleza okuthe ngqo | Iyahambelana |
Ukucaca kunye nombala wesisombululo | Cacileyo |
Izinto ezinxulumeneyo | Ukungcola ngokupheleleyo ≤1.5% Nor-nocergoline (B) ≤0.50% I-Chioronicergoline (A) ≤0.5% I-MeLUOL (C) ≤0.30% Ukungcola okungachazwanga: ≤0.30% |
Amanzi | ≤0.5% |
Intsimbi enzima | ≤20ppm |
Intsalela ekutshisweni | ≤0.05% |
Isivavanyi | 98.5%~102% |
Izinyibilikisi ezishiyekileyo | |
I-acetone | ≤1000ppm |
Diethyl ether | ≤2000ppm |
I-Ethanol | ≤1000ppm |
IMethanol | ≤1000ppm |
Toluene | ≤500ppm |
IDichloromethan | ≤100ppm |
I-Triethylamine | ≤500ppm |
Ukuqukumbela | Ukuhambelana ne-EP 5.0 |
* Ukongeza: Inkampani inokuphanda kwaye iphuhlise iimveliso ezintsha ngokwemfuno ekhethekileyo yabathengi bethu. |