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Warshada GMP waxay bixisaa tayo sare leh 99% min Triptorelin acetate cas 140194-24-7

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Warshada GMP waxay bixisaa tayo sare leh 99% min Triptorelin acetate cas 140194-24-7

Faahfaahinta alaabta:
Magaca Kiimikada: Triptorelin acetate

CAS No.: 140194-24-7

Sharaxaada Kale Ee La Xiriira

Hordhac:
Triptorelin waa gonadotropin sii daaya hormoonka (GnRH) agonist kaas oo ah xannibaad awood leh oo ka mid ah isku-darka estrogen (haweenka) waxaana loo isticmaalaa daaweynta kansarka qanjirka 'prostate'.
Waa bedelka D-tryptophan ee hadhaaga 6.

Waa daawo sababa kicinta pituitary-ga, sidaas darteed hoos u dhigista dheecaanka hormoonka luteining (LH) iyo hoormoonka stimulating follicle (FSH).
Triptorelin waa decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) iyo gonadotropin-sii daynta hormoonka agonist (GnRH agonist) loo isticmaalo sida acetate ama pamoate cusbada.

Codsiyada:
Sida kuwa kale ee GnRH agonists, triptorelin ayaa laga yaabaa in loo isticmaalo daawaynta kansarka ka jawaaba hoormoonka sida kansarka qanjirka 'prostate' ama kansarka naasaha, qaangaadhnimada hore, xaaladaha estrogen-ku-tiirsan.
(sida endometriosis ama fibroids uterine), iyo taranka la caawiyay.

Baakad:
1g/dhalo, ama sida looga baahan yahay.
Waa in lagu kaydiyaa meel qalalan, qabow iyo meel hawo leh, iska ilaali gogosha iyo qoyaanka, ka fogee oksaydhyada.

Tilmaamid

ITEM
INDEX
Astaamaha
budo crystalline cad
Assay (HPLC)
≥99%
Hal wasakh (HPLC)
≤1.0%
Halabuurka Amino Acid
± 10% ee aragtida
Waxa ku jira Peptide (N%)
≥80%
Waxyaabaha Biyaha ka kooban (Karl Fischer)
≤6.0%
Waxyaabaha Acetate (HPIC)
≤15.0%
MS(ESI)
Joogta ah
Isu-dheelitirnaanta Mass
95.0 ~ 105.0%
Wareeg gaar ah (20/D)
-65.0~-75.0°(c=0.5 1%HAc)
* Intaa waxaa dheer: Shirkaddu waxay baari kartaa oo horumarin kartaa alaabada cusub iyadoo loo eegayo baahida gaarka ah ee macaamiisheena.

 


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