Ka tukuna e te wheketere GMP te kounga teitei 99% min Triptorelin acetate cas 140194-24-7
Ka tukuna e te wheketere GMP te kounga teitei 99% min Triptorelin acetate cas 140194-24-7
Taipitopito hua:
Ingoa matū: Triptorelin acetate
Nama CAS: 140194-24-7
kupu whakataki:
Ko te Triptorelin he homone tuku gonadotropin (GnRH) agonist he aukati kaha o te whakahiato o te estrogen (i roto i nga wahine) ka whakamahia ki te rongoa i te mate pukupuku prostate matatau.
He whakakapinga D-tryptophan i te toenga 6.
He rongoa e whakaihiihi ana i te pituitary, na reira ka heke te hunanga o te taiaki luteinizing (LH) me te homoni whakaihiihi follicle (FSH).
Ko te Triptorelin he decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2) me te gonadotropin-releasing hormone agonist (GnRH agonist) i whakamahia hei tote acetate, pamoate ranei.
Nga tono:
Pērā i ērā atu agonists GnRH, ka whakamahia pea te triptorelin ki te maimoatanga o nga mate pukupuku urupare-homoni penei i te mate pukupuku prostate, te mate pukupuku uma ranei, te pakeketanga o mua, nga tikanga e whakawhirinaki ana ki te estrogen.
(pērā i te endometriosis me te fibroids uterine), me te whakawhānau āwhina.
Tapeke:
1g / pounamu, kia rite ranei ki to hiahia.
Me penapena ki te waahi maroke, hauhautanga me te hau, karohia te makuku me te makuku, kia matara atu i nga waikura.
ITEM | PANUITANGA |
Nga ahuatanga | paura tioata ma |
Whakamātautau(HPLC) | ≥99% |
Te poke kotahi (HPLC) | ≤1.0% |
Waihanga Waikawa Amino | ±10% o te ariā |
Ihirangi Peptide (N%) | ≥80% |
Ihirangi wai(Karl Fischer) | ≤6.0% |
Ihirangi Acetate (HPIC) | ≤15.0% |
MS(ESI) | Totonu |
Pauna Papatipu | 95.0~105.0% |
Tītaka Tauwhāiti (20/D) | -65.0~-75.0°(c=0.5 1%HAc) |
* I tua atu: Ka taea e te kamupene te rangahau me te whakawhanake i nga hua hou i runga i te hiahia motuhake a o taatau kiritaki. |